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BAY1125976 BAY1125976产品描述:BAY1125976是Akt1/2选择性的变构抑制剂;在10 M ATP时抑制Akt1和Akt2活性的IC50值分别为5.2 nM和18 nM。公司
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2017-07-11 |
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BAY-876 BAY-876产品描述:BAY-876是IC50为0.002 uM高选择性的GLUT1抑制剂,在体外有很好的代谢能力,在体内有高的生物利用率。公司介绍:
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2017-07-11 |
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KDM5A-IN-1 KDM5A-IN-1产品描述:KDM5A-IN-1是组蛋白去甲基化酶抑制剂。公司介绍:MedChemExpress(MCE)专注于各种抑制剂、激动剂、API及化合物
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2017-07-11 |
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Mivebresib Mivebresib产品描述:Mivebresib是BET家族的抑制剂,能够扰乱关键的转录程序在体内或者体外推动前列腺癌增长引起强的抗肿瘤特性,
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2017-07-11 |
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AZD0156 AZD0156产品描述:AZD0156是一种高效选择的,口服的ATM抑制剂,能够抑制ATM介导的信号通路,阻碍DNA损伤修复等。公司介绍:MedChe
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2017-07-11 |
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Fumarate hydratase-IN-2 Fumarate hydratase-IN-2 产品描述:.Fumarate hydratase is an enzyme of the TCA cycle and cell-permeable inhibitors(1) inh
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2017-07-11 |
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MRT68921 MRT68921产品描述:MRT68921 is the most potent inhibitor of ULK1 and ULK2, with IC50 values of 2.9 nM and 1.1 nM, respect
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2017-07-11 |
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MRT68921 (hydrochloride) MRT68921 (hydrochloride)产品描述:MRT68921 hydrochloride is the most potent inhibitor of both ULK1 and ULK2, with greate
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2017-07-11 |